Publications

2017

[479] Synthesis of CF2H-substituted pyrazolines by [3+2] cycloaddition between CF2HCHN2 and electron-deficient alkenes J. Li, X.-L. Yu, J. Cossy, S.-Y. Lv, H.-L. Zhang, F. Su, P. K. Mykhailiuk, Y. Wu Eur. J. Org. Chem. 2017, 266.

[478] A Pd-AAA approach to a-quaternary g-butyrolactones. M. Nascimento de Oliveira, J. Fournier, S. Arseniyadis, J. Cossy Org. Lett. 2017, 19, 14.

2016

[477] Synthesis of Fluoroalkyl Pyrazoles from In-Situ-Generated C2F5CHN2 and Electron-Deficient Alkenes. P.K. Mykhailiuk, A.Y. Ishchenko, V. Stepanenko, J. Cossy Eur. J. Org. Chem. 2017, 5485.

[476] Iron-Catalyzed C–C Cross-Couplings Using Organometallics. A. Guérinot, J. Cossy Top. Curr. Chem. 2016, 374, 49.

[475] Selective Tsuji-Trost type C-allylation of hydrazones: A straightforward entry into 4,5-dihydropyrazoles. H. Elhachemia, M. Cattoen, M. Cordier, J. Cossy, S. Arseniyadis, H. Ilitkie, L. El Kaïm Chem. Commun. 2016, 52, 14490-14493.

[474] Elaboration of sterically hindered delta-lactones through ring-closing metathesis: Application to the synthesis of the C1-C27 fragment of hemicalide. C. Lecourt, S. Boinapally, S. Dhambri, G. Boissonnat, C. Meyer, J. Cossy, F. Sautel, G. Massiot, J. Ardisson, G. Sorin, M.-I. Lannou J. Org. Chem. 2016, 81, 12275-12290.

[473] Iron-catalyzed synthesis of sulfur-containing heterocycles. C. Bosset, G. Lefebvre, P. Angibaud, I. Stansfield, L. Meerpoel, D. Berthelot, A. Guérinot, J. Cossy J. Org. Chem. 2016 (in press).

[472] Unexpected reactivity of trifluoromethyl diazomethane (CF3CHN2): Electrophilicity of the terminal N-atom. A. V. Arkhipov, V. V. Arkhipov, J. Cossy, V. O. Kovtunenko, P. K. Mykhailiuk Org. Lett. 2016, 18, 3406-3409.

[471] Synthetic studies toward the C14−C29 fragment of mirabalin. J. Cornil, P.-G. Echeverria, S. Reymond, P. Phansavath, V. Ratovelomanana-Vidal, A. Guérinot, J. Cossy Org. Lett. 2016, 18, 4534-4537.

[470] Synthesis of the Acyclic Carbon Skeleton of Filipin III. E. Brun, V. Bellosta, J. Cossy J. Org. Chem. 2016, 81, 8206-8221.

[469] Gold-catalyzed rearrangement of (silylcyclopropenyl)methyl ethers into (silylmethylene)cyclopropanes. F. Hiault, A. Archambeau, F. Miege, C. Meyer, J. Cossy Synthesis 2016, 48, 3165-3174.

[468] Total synthesis of putative 11-epi-lyngbouilloside aglycon. A. Kolleth, J. Gebauer, A. ElMarrouni, R. Lebeuf, C. Prévost, E. Brohan, S. Arseniyadis, J. Cossy Front. Chem, Vol 4, Article number 34, August 2016.

[467] Expanding Biohybrid-mediated Asymmetric Catalysis into the Realm of RNA. N. Duchemin, E. Benedetti, L. Bethge, S. Vonhoff, S. Klussmann, J.-J. Vasseur, J. Cossy, M. Smietana, S. Arseniyadis Chem. Commun. 2016, 52, 8604-8607.

[466] Natural Products Containing Oxygen Heterocycles—Synthetic Advances Between 1990 and 2015. J. Cossy, A. Guérinot Advances in Heterocyclic Chemistry, 2016 119, 107-142.

[465] Harnessing C–H activation of benzhydroxamates as a macrocyclization strategy: synthesis of structurally diverse macrocyclic isoquinolones. J.-P. Krieger, G. Ricci, D. Lesuisse, C. Meyer, J. Cossy Chem. Eur. J. 2016, 22, 13469-13473.

[464] Rhodium(II)-catalyzed isomerization of cyclopropenylmethyl esters into (acyloxymethylene)cyclopropanes. A. Archambeau, D.-V. Nguyen, C. Meyer, J. Cossy Chem. Eur. J. 2016, 22, 6100-6110.

[463] Design, synthesis and binding affinity evaluation of Hoechst 33258 derivatives for the development of sequence-specific DNA-based asymmetric catalysts. K. Amirbekyan, N. Duchemin, E. Benedetti, R. Joseph, A. Colon, S. A. Markarian, L. Bethge, S. Vonhoff, S. Klussmann, J. Cossy, J.-J. Vasseur, S. Arseniyadis, M. Smietana ACS Catal. 2016, 6, 3096-3105.

2015

[462] Applications in the synthesis of natural and biologically active molecules. J. Cossy in Olefin Metathesis John Wiley & Sons, Inc., Hoboken, N. J. Edited by K. Grela 2015, 287-309.

[461] Synthesis of a stereoisomer of wortmannilactone C-failure and success. A. Dittoo, D. Brandt, V. Bellosta, J. Cossy Tetrahedron 201571, 5835-5848.

[460] Beyond catalyst deactivation: cross-metathesis involving olefins containing N-heteroaromatics. K. Lafaye, C. Bosset, L. Nicolas, A. Guérinot, J. Cossy Beilstein J. Org. Chem. 2015,11, 2223-2241.

[459] Iron-catalyzed synthesis of C2 aryl and N-heteroaryl substituted tetrahydropyrans. C. Bosset, P. Angibaud, I. Stanfield, L. Meerpoel, D. Berthelot, A. Guérinot, J. Cossy J. Org. Chem. 2015, 80, 12509-12525.

[458] Total Synthesis of (+)-Cryptocaryol A Using a Prins Cyclization/Reductive Cleavage Sequence. E. Brun, V. Bellosta, J. Cossy J. Org. Chem. 2015, 80, 8668-8676.

[457] Ring contraction of 3-hydroxy-3-(trifluoromethyl)piperidines: Synthesis of 2-substituted 2-(trifluoromethyl)pyrrolidines. A. Feraldi-Xypolia, D. Gomez Pardo, J. Cossy Chem. Eur. J. 2015, 21, 12876-12880.

[456] TFA-promoted direct C–H sulfenylation at the C2 position of non-protected indoles. T. Hostier, V. Ferey, G. Ricci, D. Gomez Pardo, J. Cossy Chem. Commun. 2015, 51, 13898-13901.

[455] Synthesis of aryl sulfides: Metal-free C–H sulfenylation of electron-rich arenes. T. Hostier, V. Ferey, G. Ricci, D. Gomez Pardo, J. Cossy Org. Lett. 2015, 17, 3898-3901.

[454] Synthesis of functionalized alkylidenecyclopropanes by Ireland–Claisen rearrangement of cyclopropenylcarbinyl esters. G. Ernouf, J.-L. Brayer, B. Folléas, J.-P. Demoute, C. Meyer, J. Cossy Org. Lett. 2015, 17, 3786-3789.

[453] Cobalt-catalyzed cross-coupling of 3- and 4-iodopiperidines with Grignard reagents. L. Gonnard, A. Guérinot, J. Cossy Chem. Eur. J. 2015, 21, 12797-12803.

[452] Palladium-catalyzed phosphonylation of pyrazoles substituted by electron-withdrawing groups. Q. Huang, G. Tran, D Gomez Pardo, T. Tsuchiya, S. Hillebrand, J.-P. Vors, J. Cossy Tetrahedron 2015, 71, 7250-7259.

[451] Modular, concise, and efficient synthesis of highly functionalized 5‐fluoropyridazines by a [2+1]/[3+2]-cycloaddition sequence. G. Tran, D. Gomez Pardo, T. Tsuchiya, S. Hillebrand, J.-P. Vors, J. Cossy Org. Lett. 2015, 17, 3414-3417.

[450] Gold-catalyzed reactions of cyclopropenes. A. Archambeau, F. Miege, J. Cossy, C. Meyer PATAI’S Chemistry of Functional Groups 2015 (in press)

[449] Asymmetric transfer hydrogenation of α-amino β-keto ester hydrochlorides through dynamic kinetic resolution. P.-G. Echeverria, J. Cornil, C. Ferard, A. Guerinot, J. Cossy, P. Phansavath, V. Ratovelomanana-Vidal RSC Advances 201570, 56815-56819.

[448] Synthesis of 2-aminoindolizines by 1,3-dipolar cycloaddition of pyridinium ylides with electron-deficient ynamides. J. Brioche, C. Meyer, J. Cossy Org. Lett. 2015, 17, 2800-2803.

[447] Grignard reagents and non-precious metals: Cheap and eco-friendly reagents for developing industrial cross-couplings. A personal account. G. Cahiez, A. Moyeux, J. Cossy Adv. Synth. Catal. 2015, 357, 1983-1989.

[446] Stereoselective rearrangement of (trifluoromethyl)prolinols to enantioenriched 3-substituted 2-(trifluoromethyl)piperidines. S. Rioton, A. Orliac, Z. Antoun, R. Bidault, D. Gomez Pardo, J. Cossy Org. Lett. 2015 17, 2916-2919.

[445] Synthetic studies toward the C32-C46 segment of hemicalide. Assignment of the relative configuration of the C36-C42 subunit. S. Specklin, G. Boissonnat, C. Lecourt, G. Sorin, M.-I. Lannou, J. Ardisson, F. Sautel, G. Massiot, C. Meyer, J. Cossy Org. Lett. 2015, 17, 2446-2449.

[444] 2H-Chromenes generated by an iron(III)-complex-catalyzed allylic cyclization. L. Calmus, A. Corbu, J. Cossy Adv. Synth. Catal. 2015, 357, 1381-1386.

[443] A fast and switchable microfluidic mixer based on ultrasound-induced vaporization of perfluorocarbon. M. Bézagu, S. Arseniyadis, J. Cossy, O. Couture, M. Tanter, F. Monti, P. Tabeling Lab on a Chip 2015, 15, 2025-2029.

[442] Intramolecular cyclopropanation and C–H insertion reactions with metal carbenoids generated from cyclopropenes. A. Archambeau , F. Miege , C. Meyer, J. Cossy Acc. Chem. Res. 2015, 48, 1021-1031.

[441] Synthèse totale de molécules complexes. Evolution et nouveaux concepts. G. Massiot, J. Cossy l’Actualité Chimique 2015, février-mars, n°393-394, 39-47.

[440] Linchpin dienes: key building-blocks in the synthesis of polyenic frameworks. J. Cornil, A. Guérinot, J. Cossy Org. Biomol. Chem. 2015, 13, 4129-4142.

[439] Diastereodivergent Pictet–Spengler cyclization of bicyclic N-acyliminium ions: Controlling a quaternary stereocenter. B. de Carné-Carnavalet, J.-P. Krieger, B. Folléas, J.-L. Brayer, J.-P. Demoute, C. Meyer, J. Cossy Eur. J. Org. Chem. 2015, 1273-1282.

[438] Chemoselective synthesis of β-ketophosphonates using lithiated α-(trimethylsilyl)methylphosphonate. S. Specklin, J. Cossy J. Org. Chem. 2015, 80, 3302-3308.

[437] Iron- and indium-catalyzed reactions toward nitrogen- and oxygen-containing saturated heterocycles. J. Cornil, L. Gonnard, C. Bensoussan, A. Serra-Muns, C. Gnamm, C. Commandeur, M. Commandeur, S. Reymond, A. Guérinot, J. Cossy. Acc. Chem. Res. 2015, 48, 761-773.

[436] Heck coupling using a vinyliodo-MIDA boronate: An efficient and modular access to polyene frameworks. J. Cornil, P.-G. Echeverria, P. Phansavath, V. Ratovelomanana-Vidal, A. Guérinot, J. Cossy Org. Lett. 2015, 17, 948-951.

[435] Synthetic approach to wortmannilactone C. D. Brandt, A. Dittoo, V. Bellosta, J. Cossy Org. Lett. 2015, 17, 816-819.

[434] DNA-cellulose: An economical, fully recyclable and highly effective chiral biomaterial for asymmetric catalysis. E. Benedetti, N. Duchemin, L. Bethge, S. Vonhoff, S. Klussmann, J.-J. Vasseur, J. Cossy, M. Smietana, S. Arseniyadis Chem. Commun. 2015, 51, 6076-6079.

2014

[433] Gold-catalyzed reactions of cyclopropenes. A. Archambeau, F. Miege, J. Cossy and C. Meyer in The Chemistry of Organogold Compounds, Eds: Z. Rappoport, J. F. Liebman and I. Marek; John Wiley & Sons, Ltd: Chichester, UK, 2014, pp. 631-700

[432] Iridium–SYNPHOS-catalyzed hydrogenation through dynamic kinetic resolution of α-amino β-keto ester hydrochlorides. P.-G. Echeverria, C. Férard, J. Cornil, A. Guérinot, J. Cossy, P. Phansavath, V. Ratovelomanana-Vidal, Synlett, 2014, 2761-2764.

[431] Strength by joining methods: combining synthesis with NMR, IR, and vibrational circular dichroism spectroscopy for the determination of the relative configuration in hemicalide. E. De Gussem, W. Herrebout, S. Specklin, C. Meyer, J. Cossy, P. Bultinck Chem. Eur. J. 2014, 22, 17385-17394.

[430] Iron- and cobalt-catalyzed arylation of azetidines, pyrrolidines, and piperidines with grignard reagents. B. Barré, L. Gonnard, R. Campagne, S. Reymond, J. Marin, P. Ciapetti, M. Brellier, A. Guérinot, J. Cossy Org. Lett. 2014 16, 6160-6163.

[429] QSPR prediction of the stability constants of gadolinium(III) complexes for magnetic resonance imaging. F. Dioury, A. Duprat, G. Dreyfus, C. Ferroud, J. Cossy J. Chem. Inf. Model. 2014, 54, 2718-2731.

[428] Lewis basicity modulation of N-heterocycles: A key for successful cross-metathesis. K. Lafaye, L. Nicolas, A. Guérinot, S. Reymond, J. Cossy Org. Lett. 2014, 16, 4972-4975.

[427] Access to optically active 3-substituted piperidines by ring expansion of prolinols and derivatives. D. Gomez Pardo, J. Cossy Chemistry - A Eur. J. 201420, 4516-4525.

[426] Synthesis of LY503430 by using a selective rearrangement of β-amino alcohols induced by DAST. B. Duthion, D. Gomez Pardo, J. Cossy ARKIVOC 20143, 239-255.

[425] Lewis acid catalyzed synthesis of cyclic carbonates, precursors of 1,2- and 1,3-diols. J. Cornil, L. Gonnard, A. Guérinot, S. Reymond, J. Cossy Eur. J. Org. Chem. 2014, 4958-4962.

[424] Efficient and modular synthesis of new structurally diverse functionalized [n]paracyclophanes by a ring-distortion strategy. J.-P. Krieger, G. Ricci, D. Lesuisse, C. Meyer, J. Cossy Angew. Chem. Int. Ed 2014 53, 8705-8708.

[423] Recent developments in alkyne borylations. R. Barbeyron, E. Benedetti, J. Cossy, J.-J. Vasseur, S. Arseniyadis, M. Smietana Tetrahedron 2014 70, 8431-8452.

[422] Diastereo- and enantioselective synthesis of 1,3,5,7-tetraol structural units using a prins cyclisation/reductive cleavage sequence. E. Brun, V. Bellosta, J. Cossy Chem. Commun. 2014 50, 6718-6721.

[421] High spatiotemporal control of spontaneous reactions using ultrasound-triggered composite droplets. M. Bézagu, C. Errico, V. Chaulot-Talmon, F. Monti, M. Tanter, P. Tabeling, J. Cossy, S. Arseniyadis, O. Couture J. Am. Chem. Soc. 2014, 136, 7205-7208.

[420] Synthetic strategy toward the C44–C65 fragment of mirabalin. E. Pierre-Georges, S. Prévost, J. Cornil, C. Férard, S. Reymond, A. Guérinot, J. Cossy, V. Ratovelomanana-Vidal, P. Phansavath Org. Lett. 2014, 16, 2390-2393.

[419] Isolation, structural determination and synthetic approaches toward amphidinol 3. C. Bensoussan, N. Rival, G. Hanquet, F. Colobert, S. Reymond, J. Cossy Nat. Prod. Rep. 2014, 31, 468-488.

[418] Enantioselective synthesis and physicochemical properties of libraries of 3-amino- and 3-amidofluoropiperidines. A. Orliac, J. Routier, F. Burgat Charvillon, W. H. B. Sauer, A. Bombrun, S. S. Kulkarni, D. Gomez Pardo, J. Cossy Chemistry - A Eur. J. 2014 20, 3813-3824.

[417] Triphenylphosphine: a catalyst for the synthesis of C-aryl furanosides from furanosyl halides. L. Nicolas, P. Angibaud, I. Stansfield, L. Meerpoel, S. Reymond, J. Cossy Tetrahedron Lett. 2014, 55, 849-852.

[416] Synthesis of substituted indenones and indanones by a Suzuki-Miyaura coupling/acid-promoted cyclisation sequence. A. N. Butkevich, B. Ranieri, L. Meerpoel, I. Stansfield, P. Angibaud, A. Corbu, J. Cossy Org. Biomol. Chem. 2014, 12, 728-731.

2013

[415] Palladium-catalyzed allylic alkylation of allyl dienol carbonates. Reactivity, regioselectivity, enantioselectivity, and synthetic applications. S. Arseniyadis, J. Fournier, S. Thangavelu, O. Lozano, S. Prevost, A. Archambeau, C. Menozzi, J. Cossy Synlett 2013, 2350-2364.

[414] Palladium-catalyzed phosphonylation: Synthesis of C3, C4, and C5-phosphonylated pyrazoles. G. Tran, D. Gomez Pardo, T. Tsuchiya, S. Hillebrand, J.-P. Vors, J. Cossy Org. Lett. 2013, 15, 5550-5553.

[413] Cobalt-catalyzed diastereoselective synthesis of C furanosides. Total synthesis of (-)-isoaltholactone. L. Nicolas, E. Izquierdo, P. Angibaud, I. Stansfield, L. Meerpoel, S. Reymond, J. Cossy J. Org. Chem. 2013, 78, 11807-11814.

[412] Copper-catalysed amidation of 2-chloro-pyridines. L. Nicolas, P. Angibaud, I. Stansfield, L. Meerpoel, S. Reymond, J. Cossy RSC Advances 2013, 3, 18787-18790.

[411] Diastereoselective synthesis of the C14-C29 fragment of amphidinol 3. N. Rival, G. Hanquet, C. Bensoussan, S. Reymond, J. Cossy, F. Colobert Org. Biomol. Chem. 2013, 11, 6829-6840.

[410] Non-enzymatic acylative kinetic resolution of primary allylic amines. A. Kolleth, M. Cattoen, S. Arseniyadis, J. Cossy Chem. Commun. 2013, 49, 9338-9340.

[409] DNA vs. mirror image DNA: A universal approach to tune the absolute configuration in DNA-based asymmetric catalysis. J. Wang, E. Benedetti, L. Bethge, S. Vonhoff, S. Klussmann, J.-J. Vasseur, J. Cossy, M. Smietana, S. Arseniyadis Angew. Chem., Int. Ed. 2013, 52, 11546-11549.

[408] FeCl3·6H2O, a catalyst for the diastereoselective synthesis of cis-Isoxazolidines from N-protected δ-hydroxylamino allylic acetates. J. Cornil, A. Guérinot, S. Reymond, J. Cossy J. Org. Chem. 2013, 78, 10273-10287.

[407] Synthetic studies on hemicalide: Development of a convergent approach toward the C1-C25 fragment. G. Sorin, E. Fleury, C. Tran, E. Prost, N. Molinier, F. Sautel, G. Massiot, S. Specklin, C. Meyer, J. Cossy, M.-I. Lannou, J. Ardisson Org. Lett. 2013, 15, 4734-4737.

[406] Lyngbouilloside and related macrolides from marine cyanobacteria. A. El Marrouni, A. Kolleth, R. Lebeuf, J. Gebauer, S. Prevost, M. Heras, S. Arseniyadis, J. Cossy Natural Product Communications 2013, 8, 965-972.

[405] Iridium-catalyzed hydrogen transfer: Synthesis of substituted benzofurans, benzothiophenes, and indoles from benzyl alcohols. B. Anxionnat, D. Gomez Pardo, G. Ricci, K. Rossen, J. Cossy Org. Lett. 2013, 15, 3876-3879.

[404] Tandem Suzuki-Miyaura coupling/acid-catalyzed cyclization between vinyl ether boronates and vinyl halides: A concise approach to polysubstituted furans. A. N. Butkevich, L. Meerpoel, I. Stansfield, P. Angibaud, A. Corbu, J. Cossy Org. Lett. 2013, 15, 3840-3843.

[403] Synthesis of complex oxygenated heterocycles. L. Nicolas, A. N. Butkevich, A. Guérinot, A. Corbu, S. Reymond, J. Cossy Pure and Applied Chemistry 2013, 85, 1203-1213.

[402] Catalytic asymmetric allylic alkylation of 3-arylated piperidin-2-ones. C. Michon, A. Bethegnies, F. Capet, P. Roussel, A. de Filippis, D. Gomez-Pardo, J. Cossy, F. Agbossou-Niedercorn Eur. J. Org. Chem. 2013, 22, 4979-4985.

[401] Iron-catalyzed cross-coupling between C-bromo mannopyranoside derivatives and a vinyl Grignard reagent: toward the synthesis of the C31-C52 fragment of amphidinol 3. C. Bensoussan, N. Rival, G. Hanquet, F. Colobert, S. Reymond, J. Cossy Tetrahedron 2013, 69, 7759-7770.

[400] Synthesis of two neurokinin NK1 receptor antagonists, (+)-L-733,060 and (-)-L-733,061. A. Cochi, D. Gomez Pardo, J. Cossy Heterocycles 2012, 86, 89-116.

[399] A Sonogashira cross-coupling/5-exo-dig cyclization/ionic hydrogenation sequence: Synthesis of 4-substituted 3-azabicyclo[3.1.0]hexan-2-ones from 2-iodocyclopropanecarboxamides. B. de Carne-Carnavalet, C. Meyer, J. Cossy, B. Folleas, J.-L. Brayer, J.-P. Demoute J. Org. Chem. 2013, 78, 5794-5799.

[398] Synthesis of functionalized allenamides from ynamides by enolate claisen rearrangement. J. Brioche, C. Meyer, J. Cossy Org. Lett. 2013, 15, 1626-1629.

[397] XtalFluor-E, an efficient coupling reagent for amidation of carboxylic acids.
A. Orliac, D. Gomez Pardo, A. Bombrun Org. Lett. 2013, 15, 902-905.

[396] Synthesis of 3-hydroxypipecolic acids. A. Cochi, D. Gomez Pardo, J. Cossy
Eur. J. Org. Chem. Chem. 2013, 809-829.

[395] Chemoselective alkynylation of N-sulfonylamides versus amides and carbamates - Synthesis of tetrahydropyrazines. T. Aubineau, J. Cossy Chem. Commun. 2013, 49, 3303-3305.

[394] Palladium-catalyzed asymmetric allylic alkylation of cyclic dienol carbonates: efficient route to enantioenriched gamma-butenolides bearing an all-Carbon alpha-quaternary stereogenic center. J. Fournier, O. Lozano, C. Menozzi, S. Arseniyadis, J. Cossy Angew. Chem., Int. Ed. 2013, 52, 1257-1261.

2012

[393] Synthesis of two neurokinin NK1 receptor receptor antagonists: (+)-L-733,060 and (-)-L-733,061. A. Cochi, D. Gomez Pardo, J. Cossy Heterocycles 2012, 86, 89-116.

[392] Efficient synthesis of substituted 3-azabicyclo[3.1.0]hexan-2-ones from 2-iodocyclopropanecarboxamides using a copper-free sonogashira coupling. B. de Carne-Carnavalet, A. Archambeau, C. Meyer, J. Cossy, B. Folleas, J.-L. Brayer, J.-P. Demoute Chemistry - A Eur. J. 2012, 18, 16716-16727.

[391] Stereoselective synthesis of conjugated trienols from allylic alcohols and 1-iodo-1,3-dienes. D. Brandt, V. Bellosta, J. Cossy Org. Lett. 2012, 14, 5594-5597.

[390] Fluorine as a regiocontrol element in the ring opening of bicyclic aziridiniums. Y. H. Lam, K. N. Houk, J. Cossy, D. Gomez Pardo, A. Cochi Helv. Chim. Acta 2012, 95, 2265-2277.

[389] Two-step one-pot synthesis of benzoannulated spiroacetals by Suzuki-Miyaura coupling/acid-catalyzed spiroacetalization. A. N. Butkevich, A. Corbu, L. Meerpoel, I. Stansfield, P. Angibaud, P. Bonnet, J. Cossy, Janine Org. Lett. 2012, 14, 4998-5001.

[388] DNA as a tool for molecular discovery. M. Smietana, J.-J. Vasseur, J. Cossy, S. Arseniyadis in Modern Tools for the Synthesis of Complex Bioactive Molecules John Wiley & Sons, Inc., Hoboken, N. J. Edited by J. Cossy, S. Arseniyadis 2012, 539-555.

[387] Formal synthesis of dictyostatin and synthesis of two dictyostatin analogues. J. Gallon, J. Esteban, S. Bouzbouz, M. Campbell, S. Reymond, J. Cossy Chemistry - A Eur. J. 2012, 18, 11788-11797.

[386] First intramolecular alkylation of nitriles with primary and secondary alcohols catalyzed by iridium complexes. B. Anxionnat, D. Gomez Pardo, G. Ricci, J. Cossy Eur. J. Org. Chem. 2012, 4453-4456.

[385] Ring expansion of cyclic beta-amino alcohols induced by diethylaminosulfur trifluoride: Synthesis of cyclic amines with a tertiary fluorine at C3. B. Anxionnat, B. Robert, P. George, G. Ricci, M.-A. Perrin, D. Gomez Pardo, J. Cossy J. Org. Chem. 2012, 77, 6087-6099.

[384] Gold(I)-catalysed cycloisomerisation of 1,6-cyclopropene-enes. F. Miege, C. Meyer, J. Cossy Chemistry - A Eur. J. 2012, 18, 7810-7822.

[383] Synthesis of amines from alcohols in a nonepimerizing one-pot sequence - Synthesis of bioactive compounds: cinacalcet and dexoxadrol. C. Guerin, V. Bellosta, G. Guillamot, J. Cossy Eur. J. Org. Chem. 2012, 2990-3000.

[382] Access to optically active 3-aminopiperidines by ring expansion of prolinols: Thermodynamic versus kinetic control. A. Cochi, D. Gomez Pardo, J. Cossy Eur. J. Org. Chem. 2012, 2023-2040.

[381](E)-Dimethyl 2-oxopent-3-enylphosphonate: An excellent substrate for cross-metathesis - easy access to functionalized heterocycles. T. Cochet, D. Roche, V. Bellosta, J. Cossy Eur. J. Org. Chem. 2012, 801-809.

[380] Catalytic diastereoselective reduction of alpha,beta-epoxy and alpha,beta-aziridinyl ynones. V. Druais, C. Meyer, J. Cossy Org. Lett. 2012 14, 516-519.

[379] Total synthesis of nominal lyngbouilloside aglycon. A. ElMarrouni, R. Lebeuf, J. Gebauer, M. Heras, S. Arseniyadis, J. Cossy Org. Lett. 2012 14, 314-317.

[378] Highly Efficient Stereoselective Catalytic C(sp3)-H Insertions with Donor Rhodium Carbenoids Generated from Cyclopropenes. A. Archambeau, F. Miege, C. Meyer, J. Cossy Angew. Chem., Int. Ed. 2012 51, 11540-11544.

[377] Diastereoselective synthesis of the C17-C30 fragment of amphidinol 3. N. Rival, D. Hazelard, G. Hanquet, T. Kreuzer, C. Bensoussan, S. Reymond, J. Cossy, F. Colobert Org. Biomol. Chem. 2012 10, 9418-9428.

[376] Diastereoselective metal-catalyzed synthesis of C-aryl and C-vinyl glycosides. L. Nicolas, P. Angibaud, I. Stansfield, P. Bonnet, L. Meerpoel, S. Reymond, J. Cossy Angew. Chem., Int. Ed. 2012, 51, 11101-11104.

[375] Rhodium(III)-catalyzed allylic C-H bond amination. Synthesis of cyclic amines from omega-unsaturated N-sulfonylamines. T. Cochet, V. Bellosta, D. Roche, J.-Y. Ortholand, A. Greiner, J. Cossy Chem. Commun. 2012, 48, 10745-10747.

[374] Catalysis-based enantioselective total synthesis of myxothiazole Z, (14S)-melithiazole G and (14S)-cystothiazole F. A. Colon, T. J. Hoffman, J. Gebauer, J. Dash, J. H. Rigby, S. Arseniyadis, J. Cossy Chem. Commun. 2012, 48, 10508-10510.

[373] Kinetic resolution of propargylamines via a highly enantioselective non-enzymatic N-acylation process. A. Kolleth, S. Christoph, S. Arseniyadis, J. Cossy Chem. Commun. 2012, 48, 10511-10513.

[372] A modular and scalable one-pot synthesis of polysubstituted furans. J. Fournier, S. Arseniyadis, J. Cossy Angew. Chem., Int. Ed. 2012, 51, 7562-7566.

[371] Synthesis and evaluation of new polyenic compounds as potential PPARs modulators. D. Amans, V. Bellosta, C. Dacquet, A. Ktorza, N. Hennuyer, B. Staels, D.-H. Caignard, J. Cossy Org. Biomol. Chem. 2012, 10, 6169-6185.

[370] Spiroketals: Toward the synthesis of 39-oxobistramide K. M. Commandeur, C. Commandeur, J. Cossy Pure and Applied Chemistry 2012, 84, 1567-1574.

[369] Ritter reaction: Recent catalytic developments. A. Guérinot, S. Reymond, J. Cossy Eur. J. Org. Chem. 2012, 19-28.

2011

[368] Synthesis of a platform to access bistramides and their analogues. M. Commandeur, C. Commandeur, J. Cossy Org. Lett. 2011, 13, 6018-6021.

[367] Access to optically active 3-azido- and 3-aminopiperidine derivatives by enantioselective ring expansion of prolinols. A. Cochi, D. Gomez Pardo, J. Cossy Org. Lett. 2011, 13, 4442-4445.

[366] Monoalkylation of acetonitrile by primary alcohols catalyzed by iridium complexes. B. Anxionnat, D. Gomez Pardo, G. Ricci, J. Cossy Org. Lett. 2011, 13, 4084-4087.

[365] Peptides targeting estrogen receptor alpha-potential applications for breast cancer treatment. G. Leclercq, D. Gallo, J. Cossy, I. Laios, D. Larsimont, G. Laurent, Y. Jacquot Current Pharmaceutical Design 2011, 17, 2632-2653.

[364] N-Formylsaccharin: A new formylating agent. T. Cochet, V. Bellosta, A. Greiner, D. Roche, J. Cossy Synlett 2011, 1920-1922.

[363] FeCl3.6H2O-catalyzed synthesis of substituted cis-2,6-tetrahydropyrans from ζ-hydroxy allylic derivatives. A. Guérinot, A. Serra-Muns, C. Bensoussan, S. Reymond, J. Cossy Tetrahedron 2011, 67, 5024-5033.

[362] Mild nonepimerizing N-alkylation of amines by alcohols without transition metals. C. Guerin, V. Bellosta, G. Guillamot, J. Cossy Org. Lett. 2011, 13, 3534-3537.

[361] When cyclopropenes meet gold catalysts. F. Miege, C. Meyer, J. Cossy Beilstein J. Org. Chem. 2011, 7, 717-734.

[360] Mechanism of action of the cytotoxic macrolides amphidinolide X and J. C. Trigili, B. Pera, M. Barbazanges, J. Cossy, C. Meyer, O. Pineda, C. Rodriguez-Escrich, F. Urpi, J. Vilarrasa, J. F. Diaz, I. Barasoain ChemBioChem 2011, 12, 1027-1030.

[359] A concise approach towards the synthesis of WS75624A and WS75624B via the cross-metathesis of vinyl-functionalized thiazoles. J. Dash, B. Melillo, S. Arseniyadis, J. Cossy Tetrahedron Lett. 2011, 52, 2246-2249.

[358] Asymmetric synthesis of an antagonist of neurokinin receptors: SSR 241586. T. X. Metro, A. Cochi, D. Gomez Pardo, J. Cossy J. Org. Chem. 2011, 76, 2594-2602.

[357] Synthesis of 1,2-amino alcohols by sigmatropic rearrangements of 3-(N-tosylamino)allylic alcohol derivatives. M. Barbazanges, C. Meyer, J. Cossy, P. Turner Chemistry - A Eur. J. 2011, 17, 4480-4495.

[356] Rhodium-catalyzed cycloisomerization involving cyclopropenes: Efficient stereoselective synthesis of medium-sized heterocyclic scaffolds. F. Miege, C. Meyer, J. Cossy Angew. Chem., Int. Ed. 2011, 50, 5932-5937.

[355] Copper-free Sonogashira coupling of cyclopropyl iodides with terminal alkynes. B. de Carne-Carnavalet, A. Archambeau, C. Meyer, J. Cossy, B. Folleas, J. L. Brayer, J. P. Demoute Org. Lett. 2011, 13, 956-959.

[354] Olefin metathesis: a revolution for the synthesis of complex molecules during the 20th century. J. Cossy Actualite Chimique 2011, 70-74.

2010

[353] Silica gel-mediated rearrangement of allylic acetates. Application to the synthesis of 1,3-enynes. A. Serra-Muns, A. Guérinot, S. Reymond, J. Cossy Chem. Commun. 2010, 46, 4178-4180.

[352] Ring-rearrangement metathesis of cyclopropenes: Synthesis of heterocycles. F. Miege, C. Meyer, J. Cossy Org. Lett. 2010, 12, 248-251.

[351] Synthesis of 3-oxa- and 3-azabicyclo 4.1.0 heptanes by gold-catalyzed cycloisomerization of cyclopropenes. F. Miege, C. Meyer, J. Cossy Org. Lett. 2010, 12, 4144-4147.

[350] Rearrangement of beta-amino alcohols via aziridiniums: A review. T. X. Metro, B. Duthion, D. Gomez Pardo, J. Cossy Chem. Soc. Rev. 2010, 39, 89-102.

[349] Stereoselective synthesis of the C1-C11 and C12-C34 fragments of mycalolide A. T. J. Hoffman, A. Kolleth, J. H. Rigby, S. Arseniyadis, J. Cossy Org. Lett. 2010, 12, 3348-3351.

[348] Reduction of alkynyl alpha-Hydroxy esters: Stereoselective alpha-ketol rearrangement. T. Hameury, V. Bellosta, J. Guillemont, L. Van Hijfte, J. Cossy Eur. J. Org. Chem. 2010, 607-610.

[347] FeCl3-Catalyzed Highly Diastereoselective Synthesis of Substituted Piperidines and Tetrahydropyrans. A. Guérinot, A. Serra-Muns, C. Gnamm, C. Bensoussan, S. Reymond, J. Cossy Org. Lett. 2010, 12, 1808-1811.

[346] Synthetic efforts toward the spiroketal core of spirangien A. A. Guérinot, G. Lepesqueux, S. Sable, S. Reymond, J. Cossy J. Org. Chem. 2010, 75, 5151-5163.

[345] Ring enlargement and ring contraction induced by diethylaminosulfur trifluoride (DAST). H. Ferret, I. Dechamps, D. Gomez Pardo, L. Van Hijfte, J. Cossy Arkivoc 2010, 126-159.

[344] Two concise total syntheses of (-)-bitungolide F. A. ElMarrouni, S. R. Joolakanti, A. Colon, M. Heras, S. Arseniyadis, J. Cossy Org. Lett. 2010, 12, 4074-4077.

[343] Expedient Synthesis of a Stereoisomer of Acremolide B. A. ElMarrouni, A. Fukuda, M. Heras, S. Arseniyadis, J. Cossy J. Org. Chem. 2010, 75, 8478-8486.

[342] Enantioselective Synthesis of beta-Fluoroamines from beta-Amino Alcohols: Application to the Synthesis of LY503430. B. Duthion, D. Gomez Pardo, J. Cossy Org. Lett. 2010, 12, 4620-4623.

[341] A convergent approach toward phoslactomycins and leustroducsins. V. Druais, M. J. Hall, C. Corsi, S. V. Wendeborn, C. Meyer, J. Cossy Tetrahedron 2010, 66, 6358-6375.

[340] Efficient cyclization routes to substituted heterocyclic compounds mediated by transition-metal catalysts. J. Cossy Pure and Applied Chemistry 2010, 82, 1365-1373.

[339] Enantioselective Synthesis of SSR 241586 by Using an Organo-Catalyzed Henry Reaction. A. Cochi, T. X. Metro, D. Gomez Pardo, J. Cossy Org. Lett. 2010, 12, 3693-3695.

2009

[338] Asymmetric pentenylation of aldehydes: A new benchmark for the preparation of ethyl-substituted homoallylic alcohol. R. P. Sonawane, S. R. Joolakanti, S. Arseniyadis, J. Cossy Synlett 2009, 213-216.

[337] Highly enantioselective synthesis of linear beta-amino alcohols. T. X. Metro, D. Gomez Pardo, J. Cossy Chemistry - A Eur. J. 2009, 15, 1064-1070.

[336] A versatile route to the tulearin class of macrolactones: Synthesis of a stereoisomer of tulearin A. A. L. Mandel, V. Bellosta, D. P. Curran, J. Cossy Org. Lett. 2009, 11, 3282-3285.

[335] Straightforward synthesis of the near-infrared fluorescent voltage-sensitive dye
RH1691 and analogues thereof
. R. Lebeuf, I. Ferezou, J. Rossier, S. Arseniyadis, J. Cossy Org. Lett. 2009, 11, 4822-4825.

[334] Daucus carota-mediated reduction of cyclic 3-oxo-amines. R. Lacheretz, D. Gomez Pardo, J. Cossy Org. Lett. 2009, 11, 1245-1248.

[333] Enantioselective organocatalytic conjugate reduction of beta-azole-containing alpha,beta-unsaturated aldehydes. T. J. Hoffman, J. Dash, J. H. Rigby, S. Arseniyadis, J. Cossy Org. Lett. 2009, 11, 2756-2759.

[332] Diastereodivergent addition of allenylzincs to aryl glyoxylates. T. Hameury, J. Guillemont, L. Van Hijfte, V. Bellosta, J. Cossy Org. Lett. 2009, 11, 2397-2400.

[331] Acryloyl chloride: An excellent substrate for cross-metathesis. A one-pot sequence for the synthesis of substituted alpha,beta-unsaturated carbonyl derivatives. L. Ferrie, S. BouzBouz, J. Cossy Org. Lett. 2009, 11, 5446-5448.

[330] Rearrangement of N-alkyl 1,2-amino alcohols. Synthesis of (S)-toliprolol and (S)-propanolol. B. Duthion, T. X. Metro, D. Gomez Pardo, J. Cossy Tetrahedron 2009, 65, 6696-6706.

[329] A convergent approach toward the C1-C11 subunit of phoslactomycins and formal synthesis of phoslactomycin B. V. Druais, M. J. Hall, C. Corsi, S. V. Wendeborn, C. Meyer, J. Cossy Org. Lett. 2009, 11, 935-938.

[328] Gold-catalyzed cycloisomerizations of ene-ynamides. S. Couty, C. Meyer, J. Cossy Tetrahedron 2009, 65, 1809-1832.

[327] Convergent synthesis of the C18-C30 fragment of amphidinol 3. J. Cossy, T. Tsuchiya, S. Reymond, T. Kreuzer, F. Colobert, I. E. Marko Synlett 2009, 2706-2710.

[326] Rearrangement of beta-amino alcohols and application to the synthesis of biologically active compounds. J. Cossy, D. Gomez Pardo, C. Dumas, O. Mirguet, I. Dechamps, T. X. Metro, B. Burger, R. Roudeau, J. Appenzeller, A. Cochi Chirality 2009, 21, 850-856.

[325] Enantioselective ring expansion of prolinols: An efficient and short synthesis of 2-phenylpiperidin-3-ol derivatives and 3-hydroxypipecolic acids. A. Cochi, B. Burger, C. Navarro, D. Gomez Pardo, J. Cossy, Y. Zhao, T. Cohen Synlett 2009, 2157-2161.

[324] Iron trichloride-promoted cyclization of o-alkynylaryl isocyanates: Synthesis of 3-(chloromethylene)oxindoles. G. Cantagrel, B. de Carne-Carnavalet, C. Meyer, J. Cossy Org. Lett. 2009, 11, 4262-4265.

[323] One-pot hydrosilylation-RCM-protodesilylation: Application to the synthesis of omega-alkenyl alpha,beta-unsaturated lactones. C. Bressy, F. Bargiggia, M. Guyonnet, S. Arseniyadis, J. Cossy Synlett 2009, 565-568.

[322] Simple synthesis of conjugated all-(E)-polyenic aldehydes, ketones, and esters using chemoselective cross-metathesis and an iterative sequence of reactions: Application to the synthesis of navenone B. S. BouzBouz, C. Roche, J. Cossy Synlett 2009, 803-807.

[321] FeCl3-catalyzed Ritter reaction. Synthesis of amides. B. Anxionnat, A. Guérinot, S. Reymond, J. Cossy Tetrahedron Lett. 2009, 50, 3470-3473.

[320] Synthesis of two bioactive natural products: FR252921 and pseudotrienic acid B. D. Amans, V. Bellosta, J. Cossy Chemistry - A Eur. J. 2009, 15, 3457-3473.

[319] Synthesis of the monomeric counterpart of marinomycin A. D. Amans, L. Bareille, V. Bellosta, J. Cossy J. Org. Chem. 2009, 74, 7665-7674.

2008

[318] Une source potentielle d’anticancéreux : Les produits naturels et leurs analogues. Extraction, caractérisation, activité biologique et synthèse. J. Cossy Comptes Rendus Chimie 2008, 11, 1303-1305.

[317] A convergent total synthesis of (+)-febrifugine. B. Sieng, O. L. Ventura, V. Bellosta, J. Cossy Synlett 2008, 1216-1218.

[316] Synthetic studies toward cytostatin, a natural product inhibitor of protein phosphatase 2A. A. F. Salit, C. Meyer, J. Cossy, B. Delouvrie, L. Hennequin Tetrahedron 2008, 64, 6684-6697.

[315] Synthesis of gamma-alkylidene alpha,beta-unsaturated delta-lactones by ring-closing metathesis: Application to the synthesis of the C1-C8 subunit of biselide E. A. F. Salit, M. Barbazanges, F. Miege, M. H. Larraufie, C. Meyer, J. Cossy Synlett 2008, 2583-2586.

[314] Chemoselective reactions: Toward the synthesis of biologically active natural products with anticancer activities. S. Reymond, L. Ferrie, A. Guérinot, P. Capdevielle, J. Cossy Pure and Applied Chemistry 2008, 80, 1683-1691.

[313] Copper-catalyzed Diels-Alder reactions. S. Reymond, J. Cossy Chem. Rev. 2008, 108, 5359-5406.

[312] Migrastatin and analogues: New anti-metastatic agents. S. Reymond, J. Cossy Comptes Rendus Chimie 2008, 11, 1447-1462.

[311] Formal synthesis of leustroducsin B. J. Moise,R. P. Sonawane, C. Corsi, S. V. Wendeborn, S. Arseniyadis, J. Cossy Synlett 2008, 2617-2620.

[310] Syntheses of (S,S)-reboxetine via a catalytic stereospecific rearrangement of beta-amino alcohols. T. X. Metro, D. Gomez Pardo, J. Cossy J. Org. Chem. 2008, 73, 707-710.

[309] Synthesis of vinyl-functionalized oxazoles by olefin cross-metathesis. T. J. Hoffman, J. H. Rigby, S. Arseniyadis, J. Cossy J. Org. Chem. 2008, 73, 2400-2403.

[308] [1,2]-Wittig rearrangement of (benzyloxy)acetamides. T. Hameury, J. Guillemont, L. Van Hijfte, V. Bellosta, J. Cossy Synlett 2008, 2345-2347.

[307] Facile synthesis of the C1-C13 fragment of lyngbouilloside. J. Gebauer, S. Arseniyadis, J. Cossy Synlett 2008, 712-714.

[306] Total synthesis of cystothiazole a by microwave-assisted olefin cross-metathesis. J. Gebauer, S. Arseniyadis, J. Cossy Eur. J. Org. Chem. 2008, 2701-2704.

[305] Neopeltolide, a new promising antitumoral agent. J. Gallon, S. Reymond, J. Cossy Comptes Rendus Chimie 2008, 11, 1463-1476.

[304] Synthetic efforts toward the macrolactone core of leucascandrolide A. L. Ferrie, L Boulard, F. Pradaux, S. BouzBouz, S. Reymond, P. Capdevielle, J. Cossy J. Org. Chem. 2008, 73, 1864-1880.

[303] Total Synthesis of (+)-Dodoneine. A. Dittoo, V. Bellosta, J. Cossy Synlett 2008, 2459-2460.

[302] Synthetic efforts toward the synthesis of octalactins. M. T. Dinh, S. BouzBouz, J. L. Peglion, J. Cossy Tetrahedron 2008, 64, 5703-5710.

[301] Exiguolide, a simplified analogue of the bryostatins by Nature ? J. Cossy Comptes Rendus Chimie 2008, 11, 1477-1482.

[300] A potential source for anticancer agents: Natural products and analogues. Extraction, characterization, biological activity and synthesis. J. Cossy Comptes Rendus Chimie 2008, 11, 1303-1305.

[299] Asymmetric total synthesis of the immunosuppressant (-)-pironetin. C. Bressy, J. P. Vors, S. Hillebrand, S. Arseniyadis, J. Cossy Angew. Chem., Int. Ed. 2008, 47, 10137-10140.

[298] Synthesis of optically enriched 1,2-amino alcohols by [2,3]-Wittig rearrangements of 3-aza-allylic alcohol derivatives. M. Barbazanges, C. Meyer, J. Cossy Tetrahedron Lett. 2008, 49, 2902-2906.

[297] Total Synthesis of Amphidinolide J. M. Barbazanges, C. Meyer, J. Cossy Org. Lett. 2008, 10, 4489-4492.

2007

[296] Synthesis of 3-oxooxa- and 3-oxoazacycloalk-4-enes by ring-closing metathesis. Application to the synthesis of an inhibitor of cathepsin K. C. Taillier, T. Hameury, V. Bellosta, J. Cossy Tetrahedron 2007, 63, 4472-4490.

[295] Formal synthesis of cytostatin by a convergent approach. A. F. Salit, C. Meyer, J. Cossy Synlett 2007, 934-938.

[294] Synthesis of migrastatin and its macrolide core. S. Reymond, J. Cossy Tetrahedron 2007, 63, 5918-5929.

[293] Cross-metathesis between α-methylene-γ-butyrolactone and olefins: A dramatic additive effect. J. Moise, S. Arseniyadis, J. Cossy Org. Lett. 2007, 9, 1695-1698.

[292] Highly enantioselective synthesis of β-amino alcohols:  A catalytic version. T. X. Metro, D. Gomez Pardo, J. Cossy J. Org. Chem. 2007, 72, 6556-6561.

[291] Stereospecific rearrangement of beta-amino alcohols catalyzed by H2SO4. T. X. Metro, D. Gomez Pardo, J. Cossy Synlett 2007, 2888-2890.

[290] Studies on enol carbonate chemistry: Stereoselective construction of vicinal quaternary benzylic centers in the bis-oxindole series. C. Menozzi, P. I. Dalko, J. Cossy Heterocycles 2007, 72, 199-205.

[289] Iron-catalyzed cross-coupling of alkyl halides with alkenyl Grignard reagents. A. Guérinot, S. Reymond, J. Cossy Angew. Chem., Int. Ed. 2007, 46, 6521-6524.

[288] A concise total synthesis of melithiazole C. J. Gebauer, S. Arseniyadis, J. Cossy Org. Lett. 2007, 9, 3425-3427.

[287] Formal chemoselective synthesis of leucascandrolide A. L. Ferrie, S. Reymond, P. Capdevielle, J. Cossy Org. Lett. 2007, 9, 2461-2464.

[286] Concise total synthesis of (-)-muricatacin and (-)-iso-cladospolide B using chemoselective cross-metathesis. L. Ferrie, S. Reymond, P. Capdevielle, J. Cossy Synlett 2007, 2891-2893.

[285] Synthesis of optically active substituted 3-fluoropiperidines from prolinols by Using DAST. I. Dechamps, D. Gomez Pardo, J. Cossy Synlett 2007, 263-267.

[284] Enantioselective ring expansion of prolinols and ring-closing metathesis: formal synthesis of (-)-swainsonine. I. Dechamps, D. Gomez Pardo, J. Cossy Arkivoc 2007, 38-45.

[283] Ring expansion induced by DAST: Synthesis of substituted 3-fluoropiperidines from prolinols and 3-fluoroazepanes from 2-hydroxymethylpiperidines. I. Dechamps, D. Gomez Pardo, J. Cossy Eur. J. Org. Chem. 2007, 4224-4234.

[282] Enantioselective ring expansion of prolinol derivatives. Two formal syntheses of (-)-swainsonine. I. Dechamps, D. Gomez Pardo, J. Cossy Tetrahedron 2007, 63, 9082-9091.

[281] Synthesis of vinyl-functionalized thiazoles by cross-metathesis and tandem Stille coupling/cross-metathesis. J. Dash, S. Arseniyadis, J. Cossy Adv. Synth. & Catal. 2007, 349, 152-156.

[280] Chemoselective epoxidation of ene-ynamides: Intramolecular cyclopropanation induced by the intermediate α-oxocarbene. S. Couty, C. Meyer, J. Cossy Synlett 2007, 2819-2822.

[279] Efficient syntheses of the polyene fragments present in amphidinols. J. Cossy, T. Tsuchiya, L. Ferrie, S. Reymond, T. Kreuzer, F. Colobert, P. Jourdain, I. E. Marko Synlett 2007, 2286-2288.

[278] Stereoselective synthesis of the C53-C67 polyene fragment of amphidinol 3. F. Colobert, T. Kreuzer, J. Cossy, S. Reymond, T. Tsuchiya, L. Ferrie, I. E. Marko, P. Jourdain Synlett 2007, 2351-2354.

[277] Synthetic studies towards the marine natural product palmerolide A: synthesis of the C3-C15 and C16-C23 fragments. G. Cantagrel, C. Meyer, J. Cossy Synlett 2007, 2983-2986.

[276] Total synthesis of herbimycin A. S. Canova, V. Bellosta, A. Bigot, P. Mailliet, S. Mignani, J. Cossy Org. Lett. 2007, 9, 145-148.

[275] Ruthenium-catalyzed cross-metathesis between diallylsilanes and electron-deficient Olefins. S. BouzBouz, L. Boulard, J. Cossy Org. Lett. 2007, 9, 3765-3768.

[274] Synthesis of the C1-C13 fragment of (+)-callipeltoside A. L. Boulard, S. BouzBouz, J. M. Paris, J. Cossy Synlett 2007, 1461-1463.

[273] Highly diastereoselective addition of phenyllithium on cis-substituted C-cyclopropylaldimines. D. Belotti, N. Noujeim, J. Cossy Synlett 2007, 259-262.

[272] Stereoselective synthesis of 1,2-aminoalcohols by [2,3]-Wittig rearrangements. M. Barbazanges, C. Meyer, J. Cossy Org. Lett. 2007, 9, 3245-3248.

[271] Synthesis of an analog of mycothiazole and total synthesis of pseudotrienic acid B. D. Amans, A. Le Flohic, V. Bellosta, C. Meyer, J. Cossy Pure and Applied Chemistry 2007, 79, 677-684.

[270] An efficient and stereoselective synthesis of the monomeric counterpart of marinomycin A. D. Amans, V. Bellosta, J. Cossy Org. Lett. 2007, 9, 1453-1456.

[269] Synthesis of a promising immunosuppressant: FR252921. D. Amans, V. Bellosta, J. Cossy Org. Lett. 2007, 9, 4761-4764.

[268] A short and highly diastereoselective synthesis of verbalactone. F. Allais, M. C. Louvel, J. Cossy Synlett 2007, 451-452.

2006

[267] Synthesis of 3-oxoazacyclohept-4-enes by ring-closing metathesis. Application to the synthesis of an inhibitor of cathepsin K. C. Taillier, T. Hameury, V. Bellosta, J. Cossy Heterocycles 2006, 67, 549-554.

[266] Enantioselective diethylzinc addition to aromatic and aliphatic aldehydes using (3R,5R)-dihydroxypiperidine derivatives catalyst. R. D. Roudeau, Gomez Pardo, J. Cossy Tetrahedron 2006, 62, 2388-2394.

[265] Total synthesis of (+)-migrastatin. S. Reymond, J. Cossy Eur. J. Org. Chem. 2006, 4800-4804.

[264] Highly enantioselective synthesis of beta-amino alcohols. T. X. Metro, J. Appenzeller, D. Gomez Pardo, J. Cossy Org. Lett. 2006, 8, 3509-3512.

[263] Concise synthesis of the (+/-)-N-b-desmethyl-meso-chimonanthine. C. Menozzi, P. I. Dalko, J. Cossy. Chem. Commun. 2006, 4638-4640.

[262] Ring expansion of functionalized octahydroindoles to enantiopure cis-decahydroquinolines. M. Mena, J. Bonjoch, D. Gomez Pardo, J. Cossy J. Org. Chem. 2006, 71, 5930-5935.

[261] Reactivity of unsaturated sultones synthesized from unsaturated alcohols by ring-closing metathesis. Application to the racemic synthesis of the originally proposed structure of mycothiazole. A. Le Flohic, C. Meyer, J. Cossy Tetrahedron 2006, 62, 9017-9037.

[260] Total synthesis of (-)-spongidepsin. L. Ferrie, S. Reymond, P. Capdevielle, J. Cossy Org. Lett. 2006, 8, 3441-3443.

[259] Chemoselective cross-metathesis reaction between electron-deficient 1,3-dienes and olefins. L. Ferrie, D. Amans, S. Reymond, V. Bellosta, P. Capdevielle, J. Cossy J. Organomet. Chem. 2006, 691, 5456-5465.

[258] A short synthesis of lennoxamine via ynamides. S. Couty, C. Meyer, J. Cossy Tetrahedron Lett. 2006, 47, 767-769.

[257] Diastereoselective gold-catalyzed cycloisomerizations of ene-ynamides. S. Couty, C. Meyer, J. Cossy Angew. Chem., Int. Ed. 2006, 45, 6726-6730.

[256] Synthesis of 3-(arylmethylene)isoindolin-1-ones from ynamides by Heck-Suzuki-Miyaura domino reactions. Application to the synthesis of lennoxamine. S. Couty, B. Liegault, C. Meyer, J. Cossy Tetrahedron 2006, 62, 3882-3895.

[255] Biological evaluation of newly synthesized quinoline-5,8-quinones as Cdc25B inhibitors. J. Cossy, D. Belotti, M. Brisson, J. J. Skoko, P. Widf, J. S. Lazo Bioorg. Med. Chem. 2006, 14, 6283-6287.

[254] Generation of ketyl radical anions by photoinduced electron transfer (PET) between ketones and amines. Synthetic applications. J. Cossy, D. Belotti Tetrahedron 2006, 62, 6459-6470.

[253] Jean Rigaudy (1921-2005) - Hommage. J. Cossy Actualite Chimique 2006, 136-136.

[252] Rearrangement of homoallylic alcohols induced by DAST. S. Canova, V. Bellosta, S. Mignani, A. Bigot, J. Cossy Org. Lett. 2006, 8, 2091-2094.

[251] A short and efficient synthesis of (-)-diospongin A. C. Bressy, F. Allais, J. Cossy Synlett 2006, 3455-3456.

[250] Two approaches for efficient synthesis of (-)-colletol. S. BouzBouz, J. Cossy Tetrahedron Lett. 2006, 47, 901-904.

[249] Desymmetrization of substituted 1,3-diketones: A formal synthesis of (+)-stemoamide. N. Bogliotti, P. I. Dalko, J. Cossy Synlett 2006, 2664-2666.

[248] Free-radical approaches to stemoamide and analogues. N. Bogliotti, P. I. Dalko, J. Cossy J. Org. Chem. 2006, 71, 9528-9531.

[247] Total synthesis of pseudotrienic acid B: A bioactive metabolite from Pseudomonas sp MF 381-IODS. D. Amans, V. Bellosta, J. Cossy Angew. Chem., Int. Ed. 2006, 45, 5870-5874.

[246] Enantio- and diastereoselective allylmetalations: An easy and efficient access to the AB spiroketal of spongistatin. F. Allais, J. Cossy Org. Lett. 2006, 8, 3655-3657.

2005

[245] Hydrosilylation of terminal alkynes with alkylidene ruthenium complexes and silanes. C. Menozzi, P. I. Dalko, J. Cossy J. Org. Chem. 2005, 70, 10717-10719.

[244] In memoriam to Anne Ghosez-Giese. C. Chatgilialoglu, J. Cossy, D. P. Curran, K. B. Sharpless, and H. Yamamoto Synlett 2005, 2835-2835.

[243] A short and efficient stereoselective synthesis of the octalactin lactone using enantioselective crotyltitanations and a cross-metathesis reaction
M. T. Dinh, S. BouzBouz, J. L. Peglion, J. Cossy Synlett 2005, 2851-2853.

[242] Short synthesis of the selective Rho-kinase inhibitor Y-27632 and of its enantiomer. D. Belotti, J. L. Peglion, J. Cossy Lett. Org. Chem. 2005, 2, 634-636.

[241] Reduction of olefins using ruthenium carbene catalysts and silanes.
C. Menozzi, P. I. Dalko, J. Cossy Synlett 2005, 2449-2452.

[240] A one-pot process for the enantioselective preparation of saturated secondary alcohols from propargyl ketones under hydrogen transfer conditions.
N. Bogliotti, P. I. Dalko, J. Cossy Tetrahedron Lett. 2005, 46, 6915-6918.

[239] Regioselective synthesis of 1,2-and 1,3-diols from omega-hydroxy allyl acetates and carbonates via Pd complexes using boric acid and trialkyl borates. J. Cluzeau, P. Capdevielle, J. Cossy Tetrahedron Lett. 2005, 46, 6945-6948.

[238] Synthesis of polypropionate subunits from cyclopropanes. M. Defosseux, N. Blanchard, C. Meyer, J. Cossy Tetrahedron 2005, 61, 7632-7653.

[237] A short and enantioselective synthesis of colletodiol. L. Ferrie, P. Capdevielle, J. Cossy Synlett 2005, 1933-1935.

[236] Total synthesis of zincophorin. J. Cossy, C. Meyer, M. Defosseux, N. Blanchard Pure and Applied Chemistry 2005, 77, 1131-1137.

[235] Efficient enantioselective formal synthesis of Ro 67-8867, a NMDA 2B receptor antagonist. I. Dechamps, D. G. Pardo, P. Karoyan, J. Cossy Synlett 2005, 1170-1172.

[234] Palladium-catalyzed Suzuki-Miyaura coupling reactions involving beta,beta-dihaloenamides: Application to the synthesis of disubstituted ynamides. S. Couty, M. Barbazanges, C. Meyer, J. Cossy Synlett 2005, 905-910.

[233] Synthetic approaches and total synthesis of natural zoapatanol. C. Taillier, B. Gille, V. Bellosta, J. Cossy J. Org. Chem. 2005, 70, 2097-2108.

[232] A very short and efficient synthesis of preclamol. A. de Filippis, D. Gomez Pardo, J. Cossy Lett. Org. Chem. 2005, 2, 136-138.

[231] A radical approach for the construction of the tricyclic core of stemoamide. N. Bogliotti, P. I. Dalko, J. Cossy Synlett 2005, 349-351.

[230] A one-pot Reformatsky/cyclopropanation sequence induced by diethylzinc. M. F. Laroche, D. Belotti, J. Cossy Org. Lett. 2005, 7, 171-173.

[229] Total synthesis of ((+)(-))-mycothiazole and formal enantioselective approach. A. Le Flohic, C. Meyer, J. Cossy Org. Lett. 2005, 7, 339-342.

[228] Selective methodologies for the synthesis of biologically active piperidinic compounds. J. Cossy Chemical Records 2005, 5, 70-80.

[227] Metathesis reactions. General considerations. P. Van de Weghe, J. Eustache, J. Cossy Current Topics in Medicinal Chemistry 2005, 5, 1461-1472.

[226] Hydrogenation versus hydrogenolysis with a safe, selective and reusable catalyst: palladium black on Teflon (R). D. Belotti, G. Cantagrel, C. Combellas, J. Cossy, F. Kanoufi, S. Nunige New J. Chem. 2005, 29, 761-764.

2004

[225] Simple preparation of 3-aryl 2-piperidinones. A. de Filippis, D. Gomez Pardo, J. Cossy Synthesis 2004, 2930-2933.

[224] Palladium-catalyzed alpha-arylation of N-protected 2-piperidinones. A. de Filippis, D. Gomez Pardo, J. Cossy Tetrahedron 2004, 60, 9757-9767.

[223] Regioselective cross-metathesis reaction induced by steric hindrance. S. BouzBouz, R. Simmons, J. Cossy Org. Lett. 2004, 6, 3465-3467.

[222] Tetrafibricin: Synthesis of the C1-C13, C15-C25, and C27-C40 fragments. S. BouzBouz, J. Cossy Org. Lett. 2004, 6, 3469-3472.

[221] Stereoselective synthesis of the C15-C24 fragment of discodermolide by desymmetrization of a meso dialdehyde. S. BouzBouz, J. Cossy Synlett 2004, 2034-2036.

[220] Two successive one-pot reactions leading to the expeditious synthesis of (-)-centrolobine. L. Boulard, S. BouzBouz, J. Cossy, X. Franck, B. Figadere Tetrahedron Lett. 2004, 45, 6603-6605.

[219] Total synthesis of (+)-preussin: Control of the stereogenic centers by enantioselective allyltitanations. S. Canova, V. Bellosta, J. Cossy Synlett, 2004, 10, 1811-1813.

[218] Heck-Suzuki-Miyaura domino reactions involving ynamides. An efficient access to 3-(Arylmethylene)isoindolinones. S. Couty, B. Liegault, C. Meyer, J. Cossy Org. Lett. 2004, 6, 2511-2514.

[217] Total synthesis of zincophorin and its methyl ester. M. Defosseux, N. Blanchard, C. Meyer, J. Cossy J. Org. Chem. 2004, 69, 4626-4647.

[216] Synthesis of omega-hydroxy ketones from omega-benzyloxy Weinreb amides by using a chemoselective nucleophilic addition/birch reduction process. C. Taillier, V. Bellosta, C. Meyer, J. Cossy Org. Lett. 2004, 6, 2145-2147.

[215] Total synthesis of natural (+)-(2’S,3’R)-zoapatanol. C. Taillier, V. Bellosta, J. Cossy Org. Lett. 2004, 6, 2149-2151.

[214] Natural (5 ’-oxoheptene-1 ’ E,3 ’ E-dienyl)-5,6-dihydro-2H-pyran-2-one: total synthesis and revision of its absolute configuration. S. BouzBouz, E. de Lemos, J. Cossy, J. Saez, X. Franck, B. Figadere Tetrahedron Lett. 2004, 45, 2615-2617.

[213] Modular ligands in asymmetric synthesis. Copper-mediated cyclopropanation. D. Tepfenhart, L. Moisan, P. I. Dalko, J. Cossy Tetrahedron Lett. 2004, 45, 1781-1783.

2003

[212] Synthesis of the C14-C25 Subunit of Bafilomycin A1. F. Eustache, P. I. Dalko, J. Cossy J. Org. Chem. 2003, 68, 9994.

[211] Base effect on the palladium catalyzed a-arylation of N-benzyl-2-piperidinones. J. Cossy, A. de Filippis, D. Gomez Pardo Synlett 2003, 2171.

[210] Enantioselective monoreduction of 2-alkyl 1,3-diketones using chiral ruthenium catalysts. Synthesis of the C14-C25 fragment of bafilomycin A1. F. Eustache, P. I. Dalko, J. Cossy Tetrahedron Lett. 2003, 44, 8823.

[209] Stereoselective synthesis of polypropionate units and heterocyclic compounds by cyclopropylcarbinol ring-opening with Mercury(II) salts. C. Meyer, N. Blanchard, M. Deffosseux, J. Cossy Acc. Chem. Res. 2003, 36, 766.

[208] Solid phase synthesis of amides by the Beckmann rearrangement of ketoxime carbonates. S. His, C. Meyer, J. Cossy, G. Emeric, A. Greiner Tetrahedron Lett. 2003, 44, 8581.

[207] Synthesis of unsaturated [1,2]oxazines by using sigmatropic rearrangements and the ring-closing metathesis reaction. A. Le Flohic, C. Meyer, J. Cossy, J. R. Desmurs Tetrahedron Lett. 2003, 44, 8577.

[206] Total synthesis of zincophorin methyl ester. M. Defosseux, N. Blanchard, C. Meyer, J. Cossy Org. Lett. 2003, 5, 4037.

[205] Stereo- and enantioselective reactions. Application to the synthesis of biologically active compounds. J. Cossy, S. BouzBouz, M. Popkin Comptes Rendus Chimie 2003, 6, 547.

[204] Synthesis of indatraline using a Suzuki cross-coupling reaction and a chemoselective hydrogenation: A versatile approach. J. Cossy, D. Belotti, A. Maguer Synlett 2003, 1515.

[203] Stereoselective synthesis of the C1-C13 fragment of (+)-discodermolide using asymmetric allyltitanations. S. BouzBouz, J. Cossy Org. Lett. 2003, 5, 3029.

[202] Palladium-catalyzed intermolecular alpha-arylation of N-protected 2-piperidinones. J. Cossy, A. De Filippis, D. Gomez Pardo Org. Lett. 2003, 5, 3037.

[201] Enantioselective allyltitanations: synthesis of the proposed structures for passifloricin A. S. BouzBouz, J. Cossy Tetrahedron Lett. 2003, 44, 4471.

[200] Total synthesis of (+)-strictifolione. S. BouzBouz, J. Cossy Org. Lett. 2003, 5, 1995.

[199] Unsaturated sultones from unsaturated sulfonates: Synthesis by ring-closing metathesis and reactivity. A. Le Flohic, C. Meyer, J. Cossy, J. R. Desmurs, J. C. Galland Synlett 2003, 667.

[198] [2,3]-Wittig sigmatropic rearrangement of gamma-allyloxy-beta-enaminoesters. I. Pevet, C. Meyer, J. Cossy Synlett 2003, 663.

[197] Radical reactions. Synthesis of heterocyclic compounds. J. Cossy Bulletin de l’Union des Physiciens 2003, 97(851, Cahier 2), 29.

[196] Degradation of aldehydes to one carbon lower homologs. D. Belotti, G. Andreatta, F. Pradaux, S. BouzBouz, J. Cossy Tetrahedron Lett. 2003, 44, 3613.

[195] Tandem cross-metathesis/hydrogenation/cyclization reactions by using compatible catalysts. J. Cossy, F. Bargiggia, S. BouzBouz Org. Lett. 2003, 5, 459.

[194] Diastereoselective conjugate addition of organocuprates to chiral racemic olefinic amido esters. Formal total synthesis of paroxetine. J. Cossy, O. Mirguet, D. Gomez Pardo, J. R. Desmurs New Journal of Chemistry 2003, 27, 475.

2002

[193] A new nitrone from C2 symmetric piperidine for the synthesis of hydroxylated indolizidinone. A. Brandi, S. Cicchi, V. Paschetta, D. Gomez Pardo, J. Cossy Tetrahedron Lett. 2002, 43, 9357.

[192] Synthesis of 3-oxo oxacycloalkenes by ring closing metathesis. J. Cossy, C. Taillier, V. Bellosta Tetrahedron Lett. 2002, 43, 7263.

[191] Regioselective ring opening of epoxides by nucleophiles mediated by lithium bistrifluoromethanesulfonimide. J. Cossy, V. Bellosta, C. Hamoir, J. R. Desmurs Tetrahedron Lett. 2002, 43, 7083.

[190] Tandem reaction by using compatible catalysts: cross-metathesis reaction and hydrogenation. J. Cossy, F. C. Bargiggia, S. BouzBouz Tetrahedron Lett. 2002, 43, 6715.

[189] Formal total synthesis of (+)-methynolide. J. Cossy, D. Bauer, V. Bellosta Tetrahedron 2002, 58, 5909.

[188] Free-radical hydroxylation reactions of alkylboronates. C. Cadot, P. I. Dalko, J. Cossy, C. Ollivier, R. Chuard, P. Renaud J. Org. Chem. 2002, 67, 7193.

[187] A formal synthesis of (-)-paroxetine by enantioselective ring enlargement of a trisubstituted prolinol. J. Cossy, O. Mirguet, D. G. Pardo, J. R. Desmurs Eur. J. Org. Chem. 2002, 3543.

[186] Aromatization of enamines promoted by a catalytic amount of Pd/C. Synthesis of aromatic amines. J. Cossy, D. Belotti Org. Lett. 2002, 4, 2557.

[185] Lithium bistrifluoromethanesulfonimidate-mediated regioselective ring opening of aziridines by amines. J. Cossy, V. Bellosta, V. Alauze, J. R. Desmurs Synthesis 2002, 2211.

[184] A synthetic approach towards the C1-C9 subunit of zincophorin. J. Cossy, N. Blanchard, M. Defosseux, C. Meyer Angew. Chem., Int. Ed. 2002, 41, 2144.

[183] Stereoselective oxymercuration of cyclopropylcarbinols with anchimeric assistance by aromatic groups. J. Cossy, N. Blanchard, C. Meyer Tetrahedron Lett. 2002, 43, 1801.

[182] Olefin isomerization by a ruthenium carbenoid complex. Cleavage of allyl and homoallyl groups. C. Cadot, P. I. Dalko, J. Cossy Tetrahedron Lett. 2002, 43, 1839.

[181] Chiral titanium complexes. Synthesis of optically active unsaturated alcohols, diols, polypropionates and their use in the synthesis of biologically active compounds. J. Cossy, S. BouzBouz, F. Pradaux, C. Willis, V. Bellosta Synlett 2002, 1595.

[180] Enantioselective monoreduction of 2-alkyl-1,3-diketones mediated by chiral ruthenium catalysts. Dynamic kinetic resolution. F. Eustache, P. I. Dalko, J. Cossy Org. Lett. 2002, 4, 1263.

[179] Enantioselective Allyltitanations and Metathesis Reactions. Application to the synthesis of piperidine alkaloids (+)-sedamine and (-)-prosophylline. J. Cossy, C. Willis, V. Bellosta, S. BouzBouz J. Org. Chem. 2002, 67, 1982.

[178] Enantioselective allyltitanation. Synthesis of (-)-slaframine. J. Cossy, C. Willis, V. Bellosta, L. Saint-Jalmes Synthesis 2002, 951.

[177] Cross-metathesis reaction: direct synthesis of functionalized allylsilanes. S. BouzBouz, E. De Lemos, J. Cossy Adv. Synth. & Catal. 2002, 344, 627.

[176] Selective cyclopropylcarbinyl rearrangement of tricyclo[5.3.1.0]undecanols induced by pyridinium chlorochromate. J. Cossy, S. BouzBouz, M. Laghgar, B. Tabyaoui Tetrahedron Lett. 2002, 43, 823.

[175] Formal total synthesis of (+)-methynolide. J. Cossy, D. Bauer, V. Bellosta Synlett 2002, 715.

[174] Selective protection of spirocyclic diols. An unusual acetal opening by DIBAL-H. J. Cossy, B. Gille, V. Bellosta, A. Duprat New J. Chem. 2002, 26, 526.

[173] Modular ligands for asymmetric synthesis: enantioselective catalytic Cu(II)-mediated condensation reaction of ethyl pyruvate with Danishefsky’s diene. P. I. Dalko, L. Moisan, J. Cossy Angew. Chem., Int. Ed. 2002, 41, 625.

[172] Carbon-carbon bond forming reactions by using bistrifluoromethanesulfonimide. J. Cossy, F. Lutz, V. Alauze, C. Meyer Synlett 2002, 45.

2001

[171] A short formal synthesis of paroxetine. Diastereoselective cuprate addition to a chiral racemic olefinic amido ester. J. Cossy, O. Mirguet, D. Gomez Pardo, J. R. Desmurs Tetrahedron Lett. 2001, 42, 7805-7807.

[170] Cross-metathesis reaction. Generation of highly functionalized olefins from unsaturated alcohols. J. Cossy, S. BouzBouz, A. H. Hoveyda J. Organomet. Chem. 2001, 634, 216-221.

[169] The Iodocyclization of unsaturated dihydroxysulfonamide derivatives. N- versus O-cyclisation. J. Cossy, L. Tresnard, D. Belotti, D. Gomez Pardo Tetrahedron Lett. 2001, 42, 251-254.

[168] Synthesis of isopropenylcyclopropanes - revision of the relative configuration of cyclopropyl ketones obtained by 1,3-elimination of gamma-epoxy ketones. J. Cossy, N. Blanchard, C. Meyer Eur. J. Org. Chem. 2001, 2, 339-348.

[167] Cross-metathesis reaction. Generation of highly functionalized olefins from homoallylic alcohols. J. Cossy, S. BouzBouz J. Organomet. Chem. 2001, 327.

[166] Total Synthesis of (-)-4a,5-dihydrostreptazoline. J. Cossy, I. Pevet, C. Meyer Eur. J. Org. Chem, 2001, 2841-2850.

[165] Hydroxylation of olefins using molecular oxygen via alkylboronic esters. C. Cadot, P. I. Dalko, J. Cossy Tetrahedron Lett. 2001, 42, 1661-1663.

[164] Solid-support synthesis of 1,2-diols and g-lactones through addition of alpha-(benzyloxy)crotylindium reagents to aldehydes. J. Cossy, C. Rasamison, D. Gomez Pardo, J. A. Marshall Synlett 2001, 629-633.

[163] Diastereoselective synthesis of homopropargylic alcohols on solid support. J. Cossy, M. Defosseux, C. Meyer Synlett 2001, 815-817.

[162] Heterocyclisation of azacyanine with amines. Synthesis of new fused triazines and pyrimidine rings. M. T. Kaddachi, S. Zouari, H. Ben Ammar, J. Cossy, P. H. Kahn J. Soc. Chim. Tun. 2001, 4, 1171.

[161] Direct diastereoselective synthesis of (±)-cis and (±)-trans-4-methylpipecolic acid and derivatives. J. Cossy, D. Belotti Tetrahedron Lett. 2001, 42, 2119-2120.

[160] Efficient synthesis of substituted quinoline-5,8-quinones from 8-hydroxyquinolines by photooxygenation. J. Cossy, D. Belotti Tetrahedron Lett. 2001, 42, 4329-4331.

[159] Formal total synthesis of bisabolangelone by using a radical cyclization. J. Cossy, V. Bellosta, B. Gille Comptes Rendus de l’Académie des Sciences 2001, 4, 427-429.

[158] Formation of radicals by irradiation of alkyl halides in the presence of triethylamine. Application to the synthesis of (+)-bisabolangelone. J. Cossy, V. Bellosta, J. L. Ranaivosata, B. Gille Tetrahedron 2001, 57, 5173-5182.

[157] Composition and structural determination of the wax constituents of Jojoba oil extracted from the seeds od Simmondsia chinensis growing in Tunisia. M. T. Kaddachi, K. Mtibaa, M. Jouini, J. Cossy, P. H. Kahn J. Soc. Alg. Chim. 2001, 11, 143.

[156] Chemoselective cross-metathesis reaction. Application to the synthesis of the C1-C14 fragment of amphidinol 3. J. Cossy, S. BouzBouz Org. Lett. 2001, 3, 1451-1454.

[155] A Short Synthesis of Argatoban: a Potent Selective Thrombin Inhibitor. J. Cossy, D. Belotti Bio. Med. Chem. Lett. 2001, 11, 1989-1992.

[154] Reactivity of a-(benzoyloxy)crotylstannane with aldehydes in liquid phase and on solid support. Synthesis of substituted lactones. J. Cossy, C. Rasamison, D. Gomez Pardo J. Org. Chem. 2001, 66, 7195-7198.

[153] [2,3]-Wittig rearrangement of g-allyloxy-b-ketoesters. A new access to tetronic acids. I. Pevet, C. Meyer, J. Cossy Tetrahedron Lett. 2001, 42, 5215-5218.

[152] A short synthesis of cisapride: a gastrointestinal stimulant derived from cis-4-amino-3-methoxypiperidine. J. Cossy, J. L Molina, J. R. Desmurs Tetrahedron Lett. 2001, 42, 5713-5715.

[151] Synthesis of the C1-C12 fragment of fostriecin. J. Cossy, F. Pradaux, S. BouzBouz Org. Lett. 2001, 3, 2233-2235.

[150] Synthesis of stereotriads by oxymercuration of substitued cyclopropylcarbinols. J. Cossy, N. Blanchard, C. Meyer Org. Lett. 2001, 3, 2567-2569.

[149] Ruthenium-catalyzed asymmetric reduction of 1,3-diketones using transfer hydrogenation. J. Cossy, F. Eustache, P. Dalko Tetrahedron Lett. 2001, 42, 5005-5007.

[148] Ring expansion: Formal total synthesis of (-)-paroxetine. J. Cossy, O. Mirguet, D. Gomez Pardo, J. R. Desmurs Tetrahedron Lett. 2001, 42, 5705-5707.

[147] Efficient strategy for the synthesis of stereopentad subunits of scytophycin, discodermolide and ryfamycin S. S. BouzBouz, J. Cossy Org. Lett. 2001, 3, 3995-3998.

[146] Ring expansion. Synthesis of the velbanamine piperidine core. J. Cossy, O. Mirguet, D. Gomez Pardo Synlett 2001, 1575-1577.

[145] Enantioselective allyltitanation and cross-metathesis. Synthesis of (-)-prosophylline. J. Cossy, C. Willis, V. Bellosta Synlett 2001, 1578-1580.

2000

[144] A short and efficient synthesis of (-)-4a,5-dihydrostreptazolin. J. Cossy, I. Pevet, C. Meyer Synlett, 2000, 122-124.

[143] Enantioselective allyltitanation. Applications to the synthesis of lactone units related to compactin and mevinolin. J. Cossy, S. BouzBouz Tetrahedron Lett. 2000, 41, 3363-3366.

[142] Synthesis of amino alcohol derivatives from (L)-pyroglutamic acid on solid-phaset. J. Cossy, L. Tresnard, D. Gomez Pardo Synlett 2000, 409-411.

[141] Enantioselective synthesis of syn- and anti-1,3-diols via allyltitanation of unprotected β-hydroxy aldehydes. J. Cossy, S. BouzBouz Org. Lett. 2000, 2, 501-504.

[140] Organocopper reagents (RCu, R2CuLi) for the nucleophilic C-glycosylation of a C(2)-formyl glycal. J. Cossy, H. Rakotoarisoa Synlett 2000, 734-736.

[139] N-(2-acetoxyethyl) group as a new photolabile protecting group. J. Cossy, H. Rakotoarisoa Tetrahedron Lett. 2000, 41, 2097-2099.

[138] Metallic salts promoted radical cyclization of b-keto carboxamides and their correspnding β-enamino carboxamides. J. Cossy, A. Bouzide, C. Leblanc J. Org. Chem. 2000, 65, 7257-7265.

[137] Desymmetrization of meso aldehydes with optically active allytitanium complexes. J. Cossy, S. BouzBouz, M. Popkin Org. Lett. 2000, 2, 3449-3451.

[136] Radical carbon-carbon coupling reactions via organoboranes. C. Cadot, J. Cossy, P. Dalko J. Chem. Soc., Chem. Commun. 2000, 1017-1018.

[135] The use of TFSI-H in organic synthesis. J. Cossy, F. Lutz, V. Alauze, C. Meyer, J. R. Desmurs The Roots of Organic Development 2000, 9, 25.

[134] Troglitazone. A novel antidiabetic drug for treating insulin resistance. J. Cossy, C. Menciu, H. Rakatoarisoa, P. H. Kahn J. R. Desmurs The Roots of Organic Development 2000, 9, 9.

[133] Lewis acid-mediated nucleophilic reaction of 2-alkoxychromanes with silyl enol ethers. J. Cossy, H. Rakotoarisoa Tetrahedron Lett. 2000, 41, 7203-7205.

[132] Enantioselective allyltitanation. Efficient synthesis of the C1-C14 polyol subunit of amphotericine B. S. BouzBouz, J. Cossy Org. Lett, 2000, 2, 3975-3977.

[131] Enantioselective synthesis of propargylic alcohols by addition of enantiopure cyclopentadienyldialkoxyallyltitanium complexes to acetylenic aldehydes. F. Pradaux, S. Bouzbouz, J. Cossy, C. Ferroud, A. Falguieres Tetrahedron Lett. 2000, 41, 8877-8880.

[130] Enantioselective allyltitanation. Application to the synthesis of (+)-sedamine. J. Cossy, C. Willis, V. Bellosta, S. BouzBouz Synlett 2000, 1461-1463.

[129] The N-(2-acetoxyethyl) group as a new photolabile protecting group. J. Cossy, H. Rakotoarisoa Tetrahedron Lett. 2000, 41, 2097-2099.

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